Search Result "Bridged piperazine"


Bridged Piperazines and Piperidines as CCR1 Antagonists with Oral Activity in Models of Arthritis and Multiple Sclerosis

Journal: Letters in Drug Design & Discovery
Volume: 3 Issue: 1 Year: 2006 Page: 689-694
Author(s): Laszlo Revesz, Birgit Bollbuck, Thomas Buhl, Janet Dawson, Roland Feifel, Richard Heng, Peter Hiestand, Helmut Sparrer, Achim Schlapbach, Rudolf Waelchli, Pius Loetscher

Stereoselective Synthesis of Polysubstituted Piperazines and Oxopiperazines. Useful Building Blocks in Medicinal Chemistry

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 10 Year: 2014 Page: 1308-1316
Author(s): Alessandro Mordini,Gianna Reginato,Massimo Calamante,Lorenzo Zani

General Research Article

Novel Tri-substituted Thiazoles Bearing Piperazine Ring: Synthesis and Evaluation of their Anticancer Activity

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 5 Year: 2019 Page: 547-555
Author(s): Asaf Evrim Evren,Leyla Yurttaş,Busra Eksellı,Gulsen Akalın-Cıftcı

Research Article

Novel Piperazine Amides of Cinnamic Acid Derivatives as Tyrosinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 36-44
Author(s): Zehra Tuğçe Gür,Fatma Sezer Şenol,Suhaib Shekfeh,İlkay Erdoğan Orhan,Erden Banoğlu,Burcu Çalişkan

Synthetic Chemistry with N-Acyliminium Ions Derived from Piperazine-2,5-Diones and Related Compounds

Journal: Current Organic Synthesis
Volume: 6 Issue: 2 Year: 2009 Page: 143-168
Author(s): Carmen Avendano, Elena de la Cuesta

Synthesis of Thiophenyl Schiff Bases via Buchwald-Hartwig Coupling of Piperazines to Quinoline Motif

Journal: Current Organic Synthesis
Volume: 11 Issue: 4 Year: 2014 Page: 621-625
Author(s): Rahul V. Patel,Se Won Park

N,N-Bis(trifluoromethylquinolin-4-yl)diamino Alkanes: Synthesis and Antimalarial Activity

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 438-445
Author(s): Joseph L. Kgokong, Gilbert M. Matsabisa, Peter P. Smith, Jaco C. Breytenbach

Discovery of Novel Lead in the Group of N-substituted Piperazine Ether Derivatives with Potential Histamine H3 Receptor Activity

Journal: Medicinal Chemistry
Volume: 10 Issue: 6 Year: 2014 Page: 588-599
Author(s): Kamil J. Kuder, Marta Stachnik, Walter Schunack, Ewa Szyman ska, Katarzyna Kiec -Kononowicz

Synthesis of New Aryl(Hetaryl)-Substituted Tandospirones Under Reductive Heck Type Hydroarylations and Isoxazoline Derivatives via 1,3-Dipolar Cycloaddition Reactions with Expected Anxiolytic Activity†

Journal: Current Organic Synthesis
Volume: 10 Issue: 3 Year: 2013 Page: 481-485
Author(s): Irem Kulu, Asli Kopruceli, Gokce Goksu, Nuket Ocal

A Series of 2,4(1H,3H)-Quinazolinedione Derivatives: Synthesis and Biological Evaluation as Potential Anticancer Agents

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 1 Year: 2016 Page: 64-76
Author(s): Hulya Akgun,Demet Us Yilmaz,Rengul Cetin Atalay,Damla Gozen

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